- In the autumn-winter period, the immune system is especially susceptible to various types of attacks from pathogens.
- A weakened body malfunctions and an unpleasant phenomenon occurs, such as a cold, usually accompanied by a protracted, severe cough.
- If you do not begin to take the necessary measures to combat this symptom in time, it can provoke many complications and become chronic.
- Fortunately, today medicine offers a large selection of drugs to solve this problem, available in forms to suit every taste - tablets, capsules, suspensions.
Clenbuterol: composition and properties of the drug
Clenbuterol is a unique medicine for getting rid of all types of cough. The main properties of the syrup are a powerful expectorant effect, moisturizing the respiratory tract, softening irritated mucous membranes, and eliminating pain.
The drug helps remove signs of inflammation, activate the cells' production of new healthy mucus, and prevent the proliferation of pathogenic microorganisms.
Clenbuterol is available in the form of syrup, which is very convenient, and also has a delicate sweetish taste, as a result of which it is successfully used among pediatric patients. The drug is accompanied by official instructions (annotation) and a measuring spoon.
Clenbuterol contains original and highly effective components that provide relief to the patient in the shortest possible time:
- Clenbuterol hydrochloride is the most basic and important active ingredient with a bronchodilator effect.
- Citric acid, which creates a strongly acidic environment at the site of inflammation, destructive for many bacteria.
- Sorbitol - gives the medicine that same sweet taste, acts as a sugar substitute, which is especially important for patients who have contraindications to its use.
- Glycerin, sodium citrate, sodium benzoate, raspberry extract and other substances - as additional auxiliary components.
The components of the syrup, as a rule, do not cause hypersensitivity reactions - which, undoubtedly, is also a big advantage when choosing this medicine.
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Clenbuterol for cough: indications for use
What kind of cough can Clenbuterol relieve? Its use is indicated for:
- Asthmatic type cough (with bronchial asthma, asthmatic bronchitis).
- Allergic cough (in the form of symptomatic therapy coupled with the parallel use of suitable antihistamines).
- Non-productive forms of cough (syrup facilitates the release of mucus and accelerates its movement along the respiratory tract).
- Advanced and chronic forms of cough.
- For diseases of viral, bacterial etiology (colds, flu, pharyngitis, pneumonia, as well as laryngitis).
The syrup is especially effective in dealing with problems such as dry throat and removing large amounts of mucus from the respiratory tract.
An additional bonus is the small bactericidal and softening effect of the drug. Source: nasmorkam.net
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What are the contraindications?
The composition of the drug is distinguished by the absence of various substances that can have a negative effect on the body - it does not contain hormones, alcohols, or anesthetics.
However, there are a number of conditions in which it is better to refrain from using Clenbutarol:
- Individual hypersensitivity reactions to one or more components of the drug.
- Thyroid diseases.
- Rapid heartbeat, aortic stenosis, acute phase of myocardial infarction (the drug has a fairly high effect on the cardiovascular system).
- Pregnancy (especially its first and last trimester), lactation.
- Severe side effects.
- Clenbuterol is also contraindicated if the patient has certain eye diseases (in particular, glaucoma).
Possible side effects
Undesirable side reactions while taking the medication may occur due to failure to comply with the correct dosage or insufficiently thorough study of contraindications.
Among these types of actions, the following are most often described in clinical practice:
- Tremor of the small muscles of the body (often these are the fingers of the limbs), in severe cases - muscle cramps
- Headaches, dizziness, anxiety, nervousness (due to increased excitability of the central nervous system), general weakness, fatigue
- Sharp jumps in blood pressure, increased heart rate, cardialgia, heart rhythm disturbances (in patients with pathologies of the cardiovascular system)
- Allergic skin reactions (rashes, redness, angioedema, itching)
- Disruption of the normal functioning of the gastrointestinal tract - nausea, vomiting, dry mucous membranes
- Difficulty urinating
The list of side effects of Clenbuterol is quite extensive, so before prescribing it, specialists carefully study the patient’s medical history and life, taking into account all the individual characteristics of his body. If for some reason the drug is not suitable for the patient, it is replaced with an analogue with a similar effect, but different active components in the structure.
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How much does Clenbuterol cost: price at the pharmacy
Release form | Package | Who releases | Price |
Syrup 1 mcg/ml bottle 100 ml No. 1 | Sopharma AD, Bulgaria | 130 rub. |
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Instructions for use by adults
For adult patients and children over 12 years of age, Clenbuterol cough syrup is prescribed in a dose of 15 ml 2 times a day (preferably in the morning and evening) after meals or half an hour to an hour before meals. It is convenient to measure the amount of the drug using the measuring spoon included with it.
Before taking the medicine, it is advisable to gargle with clean water or a weak solution of chamomile to cleanse it of food particles and phlegm - otherwise the components of the syrup may not work properly and the effectiveness will be reduced.
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Clenbuterol for cough for children: dosage regimen
Clenbuterol is usually prescribed to children over 6 years of age. However, in some cases, a pediatric specialist (pediatrician) can prescribe syrup for younger patients, especially if the child has a lingering dry cough.
Most often, children willingly drink syrup because of its sweet taste and soft, enveloping consistency - this is the advantage of liquid Clenbuterol over the same medicine in tablet form.
How to properly use Clenbuterol for children and how many days should a child take it? To answer, you should carefully study the instructions for use. As a rule, single doses of the drug are as follows:
- Up to 8 months - 2.5 ml;
- From 8 months to 2 years - 5 ml;
- From 2 to 4 years - 7.5 ml;
- From 4 to 6 years - 10 ml;
- From 6 to 12 years - 12-15 ml.
For children, Clenbuterol is prescribed 2 times a day (morning, evening), before or after meals (as well as for adults).
The recommended duration of taking the drug is from three days to one week (but no more).
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Use during pregnancy and breastfeeding
Taking Clenbuterol is prohibited during pregnancy (especially in the first and last trimesters), as well as during breastfeeding (since there is a presumptive possibility of excreting the drug in the mother's breast milk.
However, no clinical studies have been conducted on this matter), as well as directly during childbirth and in the postpartum period (due to the property of inhibiting the contractions of the smooth muscles of the uterus). to the content?
Analogues: what to replace?
If there is an individual intolerance to the components of Clenbuterol, it can be replaced with another medicine with a different active substance in its composition. The most popular analogues of the drug include:
- Codelac (main component - butamirate);
- Sinekod (the main component is butamirate);
- Pertussin (includes synthetic and plant substances; the main components are thyme herb extract, potassium bromide);
- Bronchoril (main component - salbutamol);
- Berodual (main components - ipratropium bromide, fenoterol).
These medications have a good expectorant effect and are better tolerated by patients with allergic reactions to Clenbuterol.
Interaction with other drugs
- Clenbuterol for cough is strictly contraindicated to be taken with beta-blockers (metoprolol, anaprilin, etc.), since antagonism is observed with the simultaneous use of these drugs;
- When combined with sympathomimetics, a mutual increase in toxicity is observed
- When taking syrup and cardiac glycosides together, the load on the cardiovascular system sharply increases, and mutual toxicity increases.
- Clenbuterol significantly reduces the therapeutic effect of hypoglycemic drugs.
- Taking syrup and monoamine oxidase inhibitors increases the risk of intracardiac conduction disorders.
- To avoid the occurrence of such undesirable reactions, the patient should be sure to tell the attending physician about all medications he is currently taking.
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Terms of sale of the drug
Clenbuterol is dispensed strictly according to the prescription prescribed by the attending physician.
special instructions
The negative effect of Clenbuterol on the ability to drive a car has been proven. In addition, when using the medicine, you need to temporarily stop doing work that requires strong emotional stress and increased attention.
Refrain from hazardous activities due to the possibility of side effects such as dizziness, muscle tremors, decreased attention, and the patient’s performance.
How to properly store syrup?
Clenbuterol should be kept in a place protected from sunlight, out of reach of children and with moderate humidity.
The storage temperature should not exceed 25 C. The pharmaceutical product must not be frozen. The shelf life, subject to storage conditions, is up to three years.
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Finally
Clenbuterol is a fairly serious drug. It is necessary to treat its use with full responsibility.
- Before starting to take the medication, it is necessary to consult a specialist who, after collecting an anamnesis and examining the patient, will write a prescription that allows you to obtain the syrup at a pharmacy.
- The dosage is also prescribed by the attending physician - and in no case should it be taken above or below the specified amount, otherwise the risk of adverse events after an overdose significantly increases or the medicine will not be fully effective.
- If signs of intolerance appear, the use of Clenbuterol should be stopped and contact a medical professional to select another pharmaceutical product.
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Reviews about the application
It so happened that my daughter and I both got sick. Naturally, we went straight to see the pediatrician. The child, by the way, is two years old. I was diagnosed with pharyngitis, and my daughter had unilateral bronchitis. They prescribed the drug Clenbuterol, from the manufacturer Sopharma.
The dosage was as follows: 15 ml twice a day for me, 5 ml for the baby. The child, fortunately, recovered without any problems. After using it, I developed redness on my hands that were very itchy. It turned out to be an allergy.
Therefore, you need to be careful in its use. Alisa, 29 years old
We were prescribed another drug, but I was not satisfied with its cost. I asked the pharmacy for something cheaper, they offered Clenbuterol, which is suitable for both children and adults. I needed it for my 3 year old son.
The product is inexpensive and yet effective. We recovered quickly. Only the child winced at each dose. I tried it myself, it really wasn’t very tasty. In order for the child to drink, I promised to give him candy, juice, etc., cajoled him, in general.
Daria, 28 years old
The drug has different reviews, so I was wondering whether it was worth buying it. Fortunately, it's inexpensive. I decided to try taking it for my children, who were prescribed it by their therapist. I’ll say right away that I didn’t regret it.
According to the instructions, I gave them one teaspoon 2 times a day. Children have allergic reactions, but after this drug no side effects were found, which is good news.
Already on the second day they felt better, and on the fifth they were completely cured. Elena, 34 years old
We have already taken Clenbuterol 2 times. And both times he helped us out. I was diagnosed with laryngitis and cough. My husband was treated with it, as well as my son and I. The child was only one year old. The drug can be taken from 8 months. Everything is fine.
Yes, the taste is not very pleasant, however, something else is important in the medicine. This is its effectiveness, which the drug copes with with a bang. We noticed the effect already on the first day, and were treated with it for no more than a week.
Therefore, I would like to recommend him to everyone. Margarita, 30 years old
I want to say that this medicine heals gently, gradually. The bronchi relax, swelling is relieved. The effect comes quickly. And all this for a low cost. There are, of course, disadvantages. For example, a number of contraindications.
In any case, prior consultation with a doctor is necessary. I didn't have any negative consequences. A friend of mine treats her little child with it and doesn’t complain either. Overall an excellent expectorant.
Elizaveta, 27 years old
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Source: https://nasmorkam.net/klenbuterol-sirop/
Clenbuterol for children
Cough is a common symptom of illness in childhood. When it appears in children, parents strive to help their son or daughter as quickly as possible and consult a doctor. If, upon examination, a pediatrician diagnoses bronchospasm or a high risk of its occurrence, then the sick child is prescribed drugs from the group of bronchodilators. One of them is Clenbuterol. Is this remedy effective for coughs, when is it prescribed to children and in what dosage is it used?
The drug is produced by the Bulgarian companies Balkanfarma and Sopharma in two forms - syrup and tablets. Clenbuterol syrup is a viscous transparent liquid that smells like raspberries. It is sold in plastic or glass bottles, which come with a measuring cup or measuring spoon. One bottle contains 100 ml of syrup.
The solid form of Clenbuterol is a flat, white, round tablet with a dividing line (the medication is divided into halves if necessary). One box contains 50 tablets, packed in blisters of 10 pieces.
The active substance of the drug is clenbuterol in the form of hydrochloride.
In 5 ml of syrup, this compound is presented at a dosage of 5 mcg and is supplemented with citric acid, sodium citrate, glycerol, raspberry flavor, propylene glycol, sorbitol and other substances.
One tablet contains 0.02 mg of the active compound, as well as wheat starch, povidone, MCC, lactose monohydrate, magnesium stearate and silicon dioxide.
The drug is classified as a bronchodilator because it is able to influence beta-2 adrenergic receptors, which are located in the bronchi. The result of this effect is relaxation of the smooth muscles of the bronchi. In addition, the medicine has the ability to enhance the secretion of bronchial secretions and dilate blood vessels in the muscles and brain.
Clenbuterol has a very weak effect on beta-1 adrenergic receptors (and therefore it is called a selective agent), only slightly increasing the force of heart contractions. It is also noted that this medicine has the ability to slightly increase body temperature.
Clenbuterol is absorbed very well both from liquid form and from tablets. After metabolic changes in the liver, most of the drug is excreted in the urine .
The effect of taking syrup or tablets begins to appear 10-15 minutes after administration, and the maximum effect is observed 2-3 hours after taking the medicine and lasts up to 6-8 hours.
The drug is used as a symptomatic remedy for bronchial obstruction. It is used:
- For bronchitis, pneumonia and other chronic pulmonary pathologies;
- For bronchial asthma (except for an acute attack).
Sometimes a doctor prescribes syrup for tracheitis, whooping cough or laryngitis. It all depends on the course of the disease and the risks of complications in such pathologies.
Clenbuterol in syrup form is prescribed to children of any age. It is safe even for infants if prescribed by a doctor in the correct dosage. The tablet form of the drug is not used in children under 6 years of age. This is due to the ability of children to swallow tablets and to a higher concentration of the active ingredient.
It is prohibited to treat a child with Clenbuterol:
- In case of hypersensitivity to such a drug (not only to the active compound, but also to any of its other components);
- With thyrotoxicosis;
- For cardiomyopathies;
- For tachyarrhythmias.
In addition, neither syrup nor tablets are given for carbohydrate metabolism disorders, for example, malabsorption or isomaltase deficiency.
For adults, the medicine is not prescribed during breastfeeding, during myocardial infarction and during pregnancy (the medicine is allowed only in the second trimester).
In diabetes mellitus, Clenbuterol should be given with caution, since it stimulates glycogenolysis and can provoke hyperglycemia.
- When treated with Clenbuterol, negative symptoms from the central nervous system may occur, such as anxiety, headaches, sleep problems, fears, hand tremors, mental disorders, weakness and others.
- The patient's digestive system may react to this drug by causing nausea or dry mouth.
- The medicine may affect the functioning of the heart, causing heart palpitations. In addition, its use can affect blood pressure - both increase it (this effect is observed more often) and decrease it.
- Taking the medicine may provoke an allergic reaction, such as hives.
- Sometimes clenbuterol causes spasm of the blood vessels of the kidneys and bladder sphincter, which reduces the formation and excretion of urine.
The syrup is given to the child twice a day during meals. The dosage is determined by the doctor individually, taking into account the body weight and age of the small patient. Most often the medicine is prescribed as follows:
- Infants under 8 months weighing from 4 to 8 kg are given 2.5 ml of the drug.
- For a child over 8 months to 2 years old with a body weight of 8-12 kg, the medicine is prescribed in a single dosage of 5 ml.
- A child from 2 to 4 years old, whose weight is from 12 to 16 kg, is given syrup in a dose of 7.5 ml per dose.
- At the age of 4-6 years with a weight of 16 to 22 kg, a single dose of the drug is 10 ml.
- For children from 6 to 12 years old, who weigh from 22 to 35 kg, the medication is prescribed 15 ml per dose twice a day.
- At the age of over 12 years, the single dosage is also 15 ml, but the drug can be given either two or three times a day.
Depending on the tolerability of clenbuterol, the dosage may be lower.
Tablets are also prescribed twice a day, and the doctor selects a single dose of this form of the drug individually, taking into account both the age of the child and the clinical situation.
The medication is given in the morning and at night.
The average dosage of this form of medicine for children 6-12 years old is half a tablet. For a child over 12 years of age, the drug is prescribed either 1/2 tablet two or three times a day, or a whole tablet 2 times a day.
Too large a dose of Clenbuterol will increase the side effects of such a medicine and cause tachycardia, trembling of the limbs, high blood pressure and other symptoms. To treat an overdose, it is recommended to rinse the stomach, give the child activated charcoal, water-salt solutions and other necessary medications.
- Clenbuterol is often prescribed in combination with anti-inflammatory drugs, including glucocorticoid hormones.
- If the baby has a bacterial infection, this medication can be used together with antibiotics, for example, the child can be prescribed Clenbuterol and Sumamed together.
- For viral infections, the drug can be prescribed together with antiviral drugs (Arbidol, Isoprinosine, Amizon, etc.)
- The simultaneous use of beta-blockers will reduce the effect of the drug or completely eliminate it.
- The therapeutic effect of hypoglycemic drugs under the influence of Clenbuterol is reduced.
- If the drug is prescribed together with theophylline or cardiac glycosides, this increases the risk of developing arrhythmias.
- Concomitant use with other adrenergic agonists, anticholinergic drugs or tricyclic antidepressants will enhance the therapeutic effect of Clenbuterol.
- Prescription along with sympathomimetics increases the risk of side effects.
To purchase Clenbuterol at a pharmacy (any form of medication), you must first visit a doctor and get a prescription from him. The average price of 100 ml of syrup is 60-90 rubles.
It is recommended to keep a bottle of syrup or a package of tablets in a place hidden from small children and sunlight, where the temperature will exceed +25 degrees Celsius. The drug should not be frozen in liquid form. The shelf life of the tablet form and sealed bottle is 3 years, but after the first use the syrup can be stored for only one month.
There are quite a lot of positive reviews about the use of Clenbuterol in children. In them, parents note the high effectiveness of the product for dry cough. According to them, the child’s condition improves after just a few uses, and the cough becomes more moist.
The drug in syrup is also praised for its convenient form, since the sweet taste allows this medication to be given to babies without any problems, and dosing the product with a measuring cap is easy. In addition, the advantage of the drug is its affordable cost.
The disadvantages of the drug include possible side effects. Although, according to mothers, they occur very rarely, they still occur in some young patients in the form of a rash on the cheeks, nausea, headaches and other symptoms. In addition, sometimes the child does not like the sweet taste of the syrup, and the shelf life of the product after opening is very short.
You can replace Clenbuterol with bronchospasm with other medications from the same group of drugs . The doctor may prescribe:
- Ventolin. This product in the form of a dosed aerosol contains salbutamol and is approved for use in children of any age. It can be replaced by the drugs Astalin Salbutamol, Salbutamol-Teva, Salamol Eco or other aerosols with the same active ingredient.
- Berodual . The composition of this medicine includes ipratropium bromide and fenoterol. Both components relax the muscles of the bronchi. The product is produced in the form of an aerosol and solution for nebulizer inhalation. For children under six years of age, this medication is prescribed only under the supervision of a doctor. An analogue of Berodual is Ipraterol-native solution.
- Berotek . The basis of this medicine is fenoterol. The medication is produced in the form of a solution used for inhalation. Like Berodual, it can be prescribed to children under 6 years of age only under the supervision of a specialist.
For even more information about cough medicines, watch Dr. Komarovsky’s short video.
Source: https://o-krohe.ru/bronholitiki/klenbuterol/
Clenbuterol: instructions for use tablets and syrup
Latin name: Clenbuterol ATC code: R03C C13 Active ingredient: clenbuterol Manufacturer: Sopharma, Balkanpharma-
Troyan (Bulgaria)
Dispensed from the pharmacy: by prescription
Storage conditions: at temperatures up to 25°C Shelf life: 3 g.
Clenbuterol is used for cough in patients suffering from asthma, as well as for:
- Prevention and elimination of bronchospasm
- Therapy of bronchitis with concomitant bronchial obstruction syndrome.
Composition and release form
- The drug is produced in tablets and oral solution.
- Clenbuterol (tablets)
- Composition of components in 1 piece:
- Active: 20 mcg clenbuterol hydrochloride
- Related: lactose, wheat starch, CMC, Aerosil, E 572, povidone.
Round pills in the form of a flat cylinder, with a dividing strip on one of the surfaces and beveled edges.
They can be white or almost white. Packed in blisters of 10 pieces. The box contains 5 plates and a manual.
Clenbuterol (cough syrup)
Contents of components in 5 ml of drinking solution:
- Active: 5 mcg clenbuterol hydrochloride
- Structure-forming ingredients: sorbitol, glycerin, PEG, citric acid monohydrate, sodium citrate dihydrate, methyl, butyl and propyl parahydroxybenzoate, sodium benzoate, raspberry flavor, purified water.
The drug is in the form of an oral translucent solution with a viscous structure, smelling of wild raspberries. The medicine is packaged in dark-protective 100 ml bottles made of polymer material or glass. The box contains 1 bottle, manual, measuring container (spoon or cup).
Medicinal properties
Price: 388 rub.
The therapeutic effect of Clenbuterol is determined by the properties and action of its main component – the substance of the same name.
The compound has the ability to stimulate beta-adrenergic receptors for a long time. As a result, direct relaxation of the bronchial muscles is achieved.
In addition, it blocks the release of inflammatory mediators from mast cells, the main culprits of bronchospasm and the inflammatory process in them.
- Reduces swelling and eliminates congestion in the organ, reduces the degree of sputum viscosity, which helps its more active removal from the bronchi.
- The substance is capable of dilating blood vessels in the brain and skeletal muscles.
- Side effects arise mainly due to the ability to irritate the receptors of the heart muscle and thereby provoke complications in its work.
- Clenbuterol also has properties identical to anabolic drugs and can cause an increase in body temperature.
- The highest effect after taking the medication is observed 1.5-3 hours after administration, and can last for 6 to 8 hours.
The substance is absorbed in the gastrointestinal tract in full and at a high speed. A small part of the drug undergoes metabolic transformation, which is converted into 8 new compounds that do not have activity.
Excretion from the body is carried out mainly by the kidneys in several stages. About 90% of the substance is released in almost 170 hours.
Mode of application
Price: 88 rub.
- The Clenbuterol therapy regimen is prescribed by a doctor; in the absence of specific prescriptions, the recommendations for use from the manufacturer should be followed.
- Pills
- Clenbuterol can be prescribed to children exclusively from the age of 6, since the effect of the drug on younger children has not been studied.
- 6-12 years: 20 mcg per day (½ t. x 2 r.), taken in the morning and shortly before bedtime
- From 12 years old: ½ t. - up to 3 r. per day or 1 t. in the morning and before bed
Adults are allowed to take 0.5 t twice a day; in case of severe bronchospasm, the dosage can be increased to 80 mcg. For maintenance therapy, a daily dosage of 20 mcg is used.
Cough syrup
The daily amount is determined depending on the severity of the diagnosis. On average, patients over 12 years of age are recommended to drink 15 ml 2 to 3 times a day. For maintenance treatment – 10 ml twice a day.
Clenbuterol in bodybuilding and sports
Recently, the scope of use of the drug has expanded beyond therapy. In particular, the medicine is extremely popular among athletes, as it helps increase endurance and, at the same time, lose weight. But since the drug is banned by WADA, athletes use it much less often than bodybuilders.
Clenbuterol is valued by them for its ability to break down fats without affecting the muscle structure: the medicine slows down the synthesis and breakdown of protein compounds, which allows them to maintain their muscles in their original form while following a hypocaloric diet during drying.
At the same time, the drug dulls appetite, accelerates metabolic processes, and blocks the formation of new fat layers.
The drug can be used as a monocourse, but most often a combination of Clenbuterol and Thyroxine is used for drying.
The combination of these drugs makes it possible to achieve two important processes: neutralizing the process of assimilation of incoming fats and stimulating the body to process existing reserves.
The course of administration usually takes 2 weeks, since after this the body begins to become accustomed to the medicine, and, accordingly, the intensity of the action decreases. In the first days, minimal doses are used, then they are increased, bringing them to the maximum.
After finishing the treatment, another drug is used - Ketotifen to relieve the side effects of Clenbuterol.
How to take Clenbuterol for weight loss (for girls, athletes, etc.)
The drug for weight loss is used not only in the sports environment, but also by ordinary people. The course of administration is also two weeks, after which you need to take a break of 1-3 months to restore receptor sensitivity.
The dosage is determined depending on gender: the peak daily intake for men is 0.1-0.16 mg, women can take up to 0.06-0.08 mg.
It is recommended to take the tablets in the first half of the day, preferably in the morning, so as not to disturb your sleep patterns, causing insomnia. Take half an hour before breakfast or waiting two hours after it. You can drink no more than 0.05 mg at a time.
During pregnancy and breastfeeding
Studying the properties of the drug in animals revealed harmful effects on the embryo/fetus. For obvious reasons, no special studies have been conducted in pregnant women. For this reason, the use of Clenbuterol Sopharma during pregnancy is prohibited. The restriction is especially strict for the first trimester and the period before childbirth, since the medicine can provoke a strong contraction of the uterine muscles.
Breastfeeding should be avoided during treatment.
Contraindications and precautions
The medication is prohibited for use if:
- The presence of personal supersensitivity to the components present in the composition
- Thyrotoxicosis
- Acute period of MI
- Obstructive form of HCM
- Tachyarrhythmias, tachycardia
- Pheochromocytoma
- Angle-closure glaucoma
- Less than 6 years old.
Relative contraindications for which the use of Clenbuterol is possible with great precautions:
- Condition after recent MI
- Liver/kidney failure
- Myocarditis
- Disorders of cardiac contractility
- Mitral valve pathologies
- Unstable and uncompensated forms of diabetes.
- Application Notes
- After stopping taking the drug, rebound syndrome may occur, the body’s resistance to the action of the active substance.
- When treating patients with diabetes, regular monitoring of glycemic levels is required.
- Since the active substance has anabolic properties, its use can lead to weight gain, and athletes test positive for doping.
- The tablets contain wheat starch, but since its content is negligible, the drug is considered safe for patients with gluten intolerance and celiac disease.
- Clenbuterol and alcohol
- It is strictly forbidden to combine treatment with drinking alcohol, otherwise you should expect not only increased side effects, but also the development of serious complications for health and even life.
Taking alcohol together with medication can cause dangerous disturbances in the functioning of the heart, including the development of collapse. Alcoholic drinks can be taken after the medication has been completely eliminated from the body. If Clenbuterol was taken as a course, then you need to wait a break - from 3 to 30 days (depending on the medical purpose). You should check with your doctor for the exact timing.
Cross-drug interactions
During treatment with Clenbuterol, it is necessary to take into account the ability of the active component to change the effect of other drugs (in combination therapy), as well as to be affected by them:
- When taken together, the drug reduces the effectiveness of insulin and drugs with sulfonylurea derivatives.
- Sympathomimetics potentiate the effect of clenbuterol.
- When combined with beta blockers, one must take into account their ability to block or weaken the effectiveness of Clenbuterol.
- Simultaneous treatment with MAOIs and cardiac glycosides can provoke a pronounced disorder of the rhythm of the heart muscle.
Side effects and overdose
Taking Clenbuterol can provoke a negative response from the body, manifested in the form of disturbances in the internal systems:
- NS: trembling fingers, sleep disturbance (difficulty falling asleep, insomnia), causeless anxiety, headaches
- CVS: ventricular extrasystole, heart rhythm failure, decrease or increase in blood pressure, hypotension
- Gastrointestinal tract: dry mouth, nausea
- Hematopoietic organs: decreased potassium levels, hypokalemia, decreased platelet concentration (manifested by increased bleeding)
- Other conditions: skin allergies, urinary disorders.
- If these or other unmentioned individual side effects occur, you should stop taking the medication and contact your doctor.
- Taking too much of the drug causes increased adverse reactions, most severely manifested in the form of tremors of the limbs, severe anxiety, and severe tachycardia.
- Therapy
- If symptoms of intoxication appear, the medicine should be discontinued and the patient should be given symptomatic therapy.
Analogs
Analogues can be used instead of Clenubetrol only after consultation with the attending physician.
Joset
Price: (100 ml) – 207 rub., (200 ml) – 273 rub.
Multicomponent drug in the form of oral syrup. The medicine contains bromhexine, salbutamol, guaifenesin and racementol. Thanks to the combined composition, mucus liquefaction and its active removal are achieved.
The drug is used in the treatment of bronchopulmonary pathologies that are accompanied by poor sputum discharge.
Adults are recommended to drink 2 tsp three times a day. syrup, for children over 6 liters. – 1-2 tsp.
Pros:
- Breaks down the viscosity of phlegm
- Stimulates coughing
- Makes breathing easier.
Flaws:
Download instructions for use
The drug "Clenbuterol"Download instructions "Clenbuterol"
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Source: http://lekhar.ru/lekarstva/preparaty-ot-kashlja/klenbuterol-instrukcija-po-primeneniju/
Clenbuterol for cough for children - instructions for use
A child’s cough should be a reason to visit a pediatrician and conduct a quality examination (listening to the chest, taking an anamnesis).
Under certain conditions, such a symptom of respiratory system diseases can become the body’s first signal about the emergence of dangerous complications. Treatment is prescribed based on the results of diagnosis and the severity of the disease.
Recently, the drug Clenbuterol has become increasingly popular.
Indications for use
First of all, you need to figure out who this medicine can help. The instructions for use indicate that the drug has a powerful expectorant effect.
If you follow the dosage and the recommendations of specialists, the product moisturizes the mucous membrane and facilitates the discharge of sputum.
In addition, Clenbuterol is able to eliminate the inflammatory process and prevent the spread of infection to the lungs.
The medicine is prescribed to children when allergic, dry non-productive and asthmatic cough is detected.
Sometimes doctors recommend Clenbuterol to solve the problem of dry mouth that occurs as a result of high temperature and dehydration during acute respiratory viral infections and acute respiratory infections.
Composition and release form
You can buy Clenbuterol tablets and syrup at the pharmacy. For children, treatment with a liquid form of the drug is preferable. The main active ingredient of the drug is clenbuterol hydrochloride. This element moisturizes the mucous membrane and expands the bronchi.
The instructions also indicate the properties of the auxiliary components:
- sorbitol is used as a sugar substitute (important for treating a child with diabetes);
- citric acid creates an environment harmful to the proliferation of bacteria and viruses;
- Raspberry extract, glycerin, sodium benzoate give the product a pleasant taste.
The ingredients of Clenbuterol are selected in such a way as to reduce the likelihood of an allergic reaction in a child.
Operating principle
The instructions for Clenbuterol mention that syrup and tablets help fight tracheitis, whooping cough, bronchitis (acute and chronic), asthma and even emphysema.
The main purpose of the drug is to increase the lumen of the bronchi during abnormal accumulation of sputum in the respiratory tract (bronchospasm).
The description of the medicine states that the active components of Clenbuterol are capable of relaxing muscles, eliminating swelling, thinning mucus, and accelerating the elimination of phlegm. Many pediatricians recommend syrup for children to prevent the spread of pathogenic microorganisms to the lower respiratory tract due to inflammation of the bronchial walls.
Instructions for use
The dosage of Clenbuterol should be selected individually, focusing on the diagnostic results, the severity of the manifestations of the disease and the age of the patient. Typically, syrup is prescribed to children over 6 years of age, but for severe dry coughs, the medicine is also used for infants.
According to the instructions, the syrup should be drunk 2 times a day (preferably at regular intervals to ensure uniformity of effect). Single dose of the drug for a child:
- under 8 months – no more than 2.5 ml;
- up to 2 years – about 5 ml;
- 2-4 years – up to 10 ml;
- over 6 years old – 13-15 ml.
The duration of the course depends on the response of the immune system to treatment. Usually, 3-5 days are enough to soften and transform a dry cough into a productive form. In any case, therapy is not carried out longer than a week.
Side effects and contraindications
Clenbuterol rarely causes negative changes in the general condition of the child. In case of overdose, side effects are possible in the form of convulsions, headaches, increased blood pressure, allergic reactions (rash, urticaria), disturbances in the digestive system (vomiting, nausea, diarrhea), problems with urination.
According to the instructions, the drug should not be taken if a young patient has pathologies of the cardiovascular system (tachycardia, stenosis), individual intolerance to the components of the drug, diseases of the thyroid gland and glaucoma. Children suffering from hypertension and diabetes can be treated with extreme caution.
Interaction with other drugs, price and analogues
Taking Clenbuterol is not permissible during pharmacotherapy with cardiac glycosides, beta-adrenergic receptor blockers, or sympathomimetic drugs. With this interaction, the load on the heart increases significantly. That is why syrup and tablets are available only with a doctor's prescription.
Analogues of the drug are “Berodual”, “Azmaril”, “Bronholitin”. The price of syrup is 130-200 rubles, depending on the manufacturer. Shelf life – 3 years in a dry, cool (up to 25°) place.
Source: https://stop-kashel.ru/klenbuterol-ot-kashlya-dlya-detej-instruktsiya-po-primeneniyu/
Clenbuterol
Clenbuterol is a drug with adrenomimetic and bronchodilator effects.
Release form and composition
Clenbuterol is produced in the form of syrup: a colorless transparent liquid with a characteristic raspberry odor (100 ml in dark glass bottles, 1 bottle in a cardboard box with a measuring spoon included).
1 ml of syrup contains:
- Active substance: Clenbuterol – 0.001 mg (in the form of hydrochloride);
- Excipients: propyl parahydroxybenzoate – 0.05 mg, sorbitol – 280 mg, citric acid monohydrate – 7 mg, glycerol – 200 mg, propylene glycol – 100 mg, sodium citrate dihydrate – 5.8 mg, sodium benzoate – 1.2 mg, methyl parahydroxybenzoate – 0.45 mg, butyl parahydroxybenzoate – 0.05 mg, ethanol 96% – 5 mg, raspberry essence – 0.45 mg, purified water – up to 1 ml.
Pharmacological properties
Pharmacodynamics
Clenbuterol is a selective β2-adrenergic agonist. Has a rapid bronchodilator effect.
The mechanism of influence is due to the specific stimulation of β2 adrenergic receptors of smooth muscles.
Binding with them activates the enzyme adenylate cyclase, which results in an increase in the intracellular concentration of cyclic adenosine monophosphate and activation of protein kinase A.
Thus, myosin is deprived of the ability to connect with actin, which causes relaxation of the bronchi.
Clenbuterol, by stimulating the cells of the bronchial mucosa, increases expectoration. When used in therapeutic doses, the drug has no effect on blood pressure and heart rate.
Pharmacokinetics
Clenbuterol is absorbed from the gastrointestinal tract relatively quickly.
Binds to plasma proteins at a level of 89–98%.
Biological T1/2 (half-life) – 3.5 hours. It is excreted primarily in the form of sulfoconjugated derivatives by the kidneys.
Indications for use
According to the instructions, Clenbuterol is prescribed for the treatment of bronchial asthma and chronic obstructive pulmonary disease (COPD).
Contraindications
- Myocardial infarction (in the acute period);
- Tachyarrhythmia;
- Hypertrophic obstructive cardiomyopathy;
- Thyrotoxicosis;
- Pheochromocytoma;
- Angle-closure glaucoma;
- Pregnancy (I and III trimester) and the period of breastfeeding (lactation);
- Age up to 6 years;
- Hypersensitivity to the components of the drug.
Clenbuterol is prescribed with caution immediately after a myocardial infarction, as well as in patients with heart rhythm disturbances, renal and liver failure, myocarditis, hypokalemia, mitral valve defects, unstable or uncompensated diabetes.
Instructions for use of Clenbuterol: method and dosage
Clenbuterol syrup is taken orally.
The daily dose is determined by age:
- Children 6-12 years old (body weight 22-35 kg) – 0.015 mg;
- Adults and children over 12 years of age: 0.02-0.04 mg.
- The frequency of administration is 2 times a day.
- Maintenance dose – 0.01 mg 2 times a day.
- On average, Clenbuterol is used for 2-3 days (until the acute symptoms of the disease subside).
The duration of maintenance treatment is up to 7 days. Longer therapy is possible after consultation with a doctor.
Side effects
When using Clenbuterol, the following side effects may develop:
- Cardiovascular system: increase or decrease in blood pressure, angina pain, tachycardia, ventricular extrasystole;
- Central nervous system: headache, anxiety;
- Muscular system: fine muscle tremors;
- Genitourinary system: urinary disturbance;
- Circulatory system: hypoglycemia, thrombocytopenia;
- Gastrointestinal tract: diarrhea, gastritis, nausea, dry mouth;
- Mucous membranes and skin: facial swelling, skin rash, urticaria.
These adverse reactions usually resolve within 7-14 days without stopping therapy.
Overdose
Main symptoms: tachycardia, headache, increased sweating, tremor of fingers; in especially severe cases - convulsions, collapse and coma.
Therapy: withdrawal of Clenbuterol (for any degree of overdose), gastric lavage, intake of activated charcoal, forced diuresis, symptomatic treatment. Use of the drug in excess of recommended doses may cause a worsening of bronchial asthma, which requires immediate medical attention and, if necessary, hospitalization.
special instructions
Clenbuterol syrup contains so-called parabens as auxiliary components: propyl parahydroxybenzoate and methyl parahydroxybenzoate, which can lead to the development of urticaria and contact dermatitis (delayed allergic reactions). In rare cases, immediate allergic reactions (bronchospasm) may occur.
- Glycerol, which is part of the syrup, in high doses can cause stomach irritation, diarrhea and headache.
- 1 ml of Clenbuterol contains 5 mg of 96% ethanol, which is dangerous for patients with alcoholism, liver disease, epilepsy, diseases or brain damage, as well as for children and pregnant women.
- Due to the presence of sorbitol in the drug, it should not be taken by patients with congenital fructose intolerance.
- Clenbuterol may enhance the effects of other medications.
Impact on the ability to drive vehicles and complex mechanisms
In the first days of therapy, the drug may cause anxiety and slight tremor, which requires increased caution when driving and operating equipment.
Use during pregnancy and lactation
- Clenbuterol is not prescribed in the first and third trimesters of pregnancy and during lactation.
- In the second trimester of pregnancy, the use of the drug is permitted, but it is recommended to give preference to the inhaled form.
- If it is necessary to use the drug during lactation, breastfeeding should be interrupted or clenbuterol should be used in the form of inhalations.
Use in childhood
Clenbuterol therapy is contraindicated in patients under 6 years of age.
For impaired renal function
Clenbuterol for renal failure should be used under medical supervision.
For liver dysfunction
Clenbuterol for liver failure should be used under medical supervision.
Drug interactions
When Clenbuterol is used simultaneously with certain medications, undesirable effects may occur:
- Beta-blockers: suppression of the action of Clenbuterol, risk of developing bronchospasm;
- Beta-adrenergic agonists, theophylline and anticholinergics: enhancing their action and side effects;
- Hypoglycemic drugs: reduction of their effect;
- Halogenated hydrocarbons for anesthesia (during manipulations and interventions): increased risk of arrhythmias;
- Monoamine oxidase inhibitors (tricyclic antidepressants): heart rhythm disturbances.
The simultaneous use of Clenbuterol with cardiac glycosides and diuretics is possible, but with periodic monitoring of serum electrolytes.
Analogs
Analogs of Clenbuterol are: Clenbuterol Sopharma, Saltos, Stanozolol.
Terms and conditions of storage
Store out of reach of children at temperatures up to 25 °C.
Shelf life – 3 years.
Conditions for dispensing from pharmacies
Dispensed by prescription.
Reviews about Clenbuterol
According to reviews, Clenbuterol is an inexpensive drug that has a quick effect. Disadvantages include a large list of contraindications and the possibility of side effects. It is also noted as a disadvantage that the syrup can be taken for no more than a month after opening the package.
Price for Clenbuterol in pharmacies
The approximate price for Clenbuterol (1 bottle of 100 ml) is 65–85 rubles.
Source: https://www.neboleem.net/clenbuterol.php